Benzoxazinone synthesis via Passerini-Smiles couplings

Elodie Martinand-Lurin; Laurent El Kaïm; Laurence Grimaud

doi:10.1016/j.tetlet.2014.07.088

Benzoxazinone synthesis via Passerini-Smiles couplings

Elodie Martinand-Lurin, Laurent El Kaïm, Laurence Grimaud

Research output: Contribution to journal › Article › peer-review

Abstract

Benzoxazinones are easily prepared using Passerini-Smiles couplings of o-nitrophenol derivatives. Palladium-catalyzed flow-hydrogenation of adducts gives aniline derivatives that cyclize into benzoxazinones on treatment with trifluoroacetic acid.

Original language	English
Pages (from-to)	5144-5146
Number of pages	3
Journal	Tetrahedron Letters
Volume	55
Issue number	37
DOIs	https://doi.org/10.1016/j.tetlet.2014.07.088
Publication status	Published - 10 Sept 2014
Externally published	Yes

Keywords

Benzoxazinone
Hydrogenation
Isocyanide
Multicomponent reaction
Passerini-Smiles

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10.1016/j.tetlet.2014.07.088

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@article{e93857ecb0b745fe876854e4565f5a06,

title = "Benzoxazinone synthesis via Passerini-Smiles couplings",

abstract = "Benzoxazinones are easily prepared using Passerini-Smiles couplings of o-nitrophenol derivatives. Palladium-catalyzed flow-hydrogenation of adducts gives aniline derivatives that cyclize into benzoxazinones on treatment with trifluoroacetic acid.",

keywords = "Benzoxazinone, Hydrogenation, Isocyanide, Multicomponent reaction, Passerini-Smiles",

author = "Elodie Martinand-Lurin and \{El Ka{\"i}m\}, Laurent and Laurence Grimaud",

year = "2014",

month = sep,

day = "10",

doi = "10.1016/j.tetlet.2014.07.088",

language = "English",

volume = "55",

pages = "5144--5146",

journal = "Tetrahedron Letters",

issn = "0040-4039",

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TY - JOUR

T1 - Benzoxazinone synthesis via Passerini-Smiles couplings

AU - Martinand-Lurin, Elodie

AU - El Kaïm, Laurent

AU - Grimaud, Laurence

PY - 2014/9/10

Y1 - 2014/9/10

N2 - Benzoxazinones are easily prepared using Passerini-Smiles couplings of o-nitrophenol derivatives. Palladium-catalyzed flow-hydrogenation of adducts gives aniline derivatives that cyclize into benzoxazinones on treatment with trifluoroacetic acid.

AB - Benzoxazinones are easily prepared using Passerini-Smiles couplings of o-nitrophenol derivatives. Palladium-catalyzed flow-hydrogenation of adducts gives aniline derivatives that cyclize into benzoxazinones on treatment with trifluoroacetic acid.

KW - Benzoxazinone

KW - Hydrogenation

KW - Isocyanide

KW - Multicomponent reaction

KW - Passerini-Smiles

U2 - 10.1016/j.tetlet.2014.07.088

DO - 10.1016/j.tetlet.2014.07.088

M3 - Article

AN - SCOPUS:84908249141

SN - 0040-4039

VL - 55

SP - 5144

EP - 5146

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 37

ER -

Benzoxazinone synthesis via Passerini-Smiles couplings

Abstract

Keywords

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