Copper-catalyzed direct amination of halo(hetero)arenes with sodium azide as the amino source

S. Messaoudi; J. D. Brion; M. Alami

doi:10.2174/157019311797440236

Copper-catalyzed direct amination of halo(hetero)arenes with sodium azide as the amino source

S. Messaoudi
, J. D. Brion
, M. Alami

Université Paris-Saclay

Research output: Contribution to journal › Article › peer-review

18 Citations (Scopus)

Abstract

In the synthesis of primary (hetero)aryl amines through copper-catalysis, the ammonia surrogates or aqueous ammonia nucleophilic partners can be replaced by sodium azide. Recent efforts in copper-mediated transformation of (hetero)aryl halides to (hetero) aryl amines using azide anion as the amino source are discussed in these highlights.

Original language	English
Pages (from-to)	448-454
Number of pages	7
Journal	Mini-Reviews in Organic Chemistry
Volume	8
Issue number	4
DOIs	https://doi.org/10.2174/157019311797440236
Publication status	Published - 1 Jan 2011
Externally published	Yes

Keywords

Amination
Aminoheterocycles
Anilines
Copper
Sodium azide

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10.2174/157019311797440236

Cite this

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abstract = "In the synthesis of primary (hetero)aryl amines through copper-catalysis, the ammonia surrogates or aqueous ammonia nucleophilic partners can be replaced by sodium azide. Recent efforts in copper-mediated transformation of (hetero)aryl halides to (hetero) aryl amines using azide anion as the amino source are discussed in these highlights.",

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AU - Messaoudi, S.

AU - Brion, J. D.

AU - Alami, M.

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Y1 - 2011/1/1

N2 - In the synthesis of primary (hetero)aryl amines through copper-catalysis, the ammonia surrogates or aqueous ammonia nucleophilic partners can be replaced by sodium azide. Recent efforts in copper-mediated transformation of (hetero)aryl halides to (hetero) aryl amines using azide anion as the amino source are discussed in these highlights.

AB - In the synthesis of primary (hetero)aryl amines through copper-catalysis, the ammonia surrogates or aqueous ammonia nucleophilic partners can be replaced by sodium azide. Recent efforts in copper-mediated transformation of (hetero)aryl halides to (hetero) aryl amines using azide anion as the amino source are discussed in these highlights.

KW - Amination

KW - Aminoheterocycles

KW - Anilines

KW - Copper

KW - Sodium azide

U2 - 10.2174/157019311797440236

DO - 10.2174/157019311797440236

M3 - Article

AN - SCOPUS:80053483890

SN - 1570-193X

VL - 8

SP - 448

EP - 454

JO - Mini-Reviews in Organic Chemistry

JF - Mini-Reviews in Organic Chemistry

IS - 4

ER -

Copper-catalyzed direct amination of halo(hetero)arenes with sodium azide as the amino source

Abstract

Keywords

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