Solvent-free amination of heteroaromatic chlorides

Erwan Le Gall; Stéphane Sengmany; Corinne Gosmini; Jacques Périchon; Pascal Retailleau

doi:10.2174/157017808783743885

Solvent-free amination of heteroaromatic chlorides

Erwan Le Gall
, Stéphane Sengmany
, Corinne Gosmini
, Jacques Périchon
, Pascal Retailleau

Université de PARIS XII
Institut de Chimie des Substances Naturelles

Research output: Contribution to journal › Article › peer-review

Abstract

The coupling of 5-membered heterocyclic amines such as pyrazole and imidazole derivatives with heteroaromatic chlorides like 4,7-dichloroquinoline, 2-chlorobenzoxazole and 2-chlorobenzothiazole has been realized in good yields using very simple solvent-free conditions.

Original language	English
Pages (from-to)	120-124
Number of pages	5
Journal	Letters in Organic Chemistry
Volume	5
Issue number	2
DOIs	https://doi.org/10.2174/157017808783743885
Publication status	Published - 1 Mar 2008
Externally published	Yes

Keywords

Amination
Heteroaromatic chlorides
Solvent-free reaction

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title = "Solvent-free amination of heteroaromatic chlorides",

abstract = "The coupling of 5-membered heterocyclic amines such as pyrazole and imidazole derivatives with heteroaromatic chlorides like 4,7-dichloroquinoline, 2-chlorobenzoxazole and 2-chlorobenzothiazole has been realized in good yields using very simple solvent-free conditions.",

keywords = "Amination, Heteroaromatic chlorides, Solvent-free reaction",

author = "\{Le Gall\}, Erwan and St{\'e}phane Sengmany and Corinne Gosmini and Jacques P{\'e}richon and Pascal Retailleau",

year = "2008",

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doi = "10.2174/157017808783743885",

language = "English",

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journal = "Letters in Organic Chemistry",

issn = "1570-1786",

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T1 - Solvent-free amination of heteroaromatic chlorides

AU - Le Gall, Erwan

AU - Sengmany, Stéphane

AU - Gosmini, Corinne

AU - Périchon, Jacques

AU - Retailleau, Pascal

PY - 2008/3/1

Y1 - 2008/3/1

N2 - The coupling of 5-membered heterocyclic amines such as pyrazole and imidazole derivatives with heteroaromatic chlorides like 4,7-dichloroquinoline, 2-chlorobenzoxazole and 2-chlorobenzothiazole has been realized in good yields using very simple solvent-free conditions.

AB - The coupling of 5-membered heterocyclic amines such as pyrazole and imidazole derivatives with heteroaromatic chlorides like 4,7-dichloroquinoline, 2-chlorobenzoxazole and 2-chlorobenzothiazole has been realized in good yields using very simple solvent-free conditions.

KW - Amination

KW - Heteroaromatic chlorides

KW - Solvent-free reaction

U2 - 10.2174/157017808783743885

DO - 10.2174/157017808783743885

M3 - Article

AN - SCOPUS:46149105016

SN - 1570-1786

VL - 5

SP - 120

EP - 124

JO - Letters in Organic Chemistry

JF - Letters in Organic Chemistry

IS - 2

ER -

Solvent-free amination of heteroaromatic chlorides

Abstract

Keywords

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