The Metabolic Fate of isoCombretastatin A-4 in Human Liver Microsomes: Identification, Synthesis and Biological Evaluation of Metabolites

Mohamed Ali Soussi, Silvio Aprile, Samir Messaoudi, Olivier Provot, Erika DelGrosso, Jérôme Bignon, Joëlle Dubois, Jean Daniel Brion, Giorgio Grosa, Mouad Alami

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Pages (from-to)1781-1788
Number of pages8
JournalChemMedChem
Volume6
Issue number10
DOIs
Publication statusPublished - 4 Oct 2011
Externally publishedYes

Keywords

  • Anticancer agents
  • Cytotoxicity
  • Drug metabolism
  • Isocombretastatin A-4
  • Tubulin

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