Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues

Laurent El Kaïm; Laurence Grimaud; Patil Pravin

doi:10.1021/ol202974w

Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues

Laurent El Kaïm
, Laurence Grimaud
, Patil Pravin

Unité Chimie et Procédés

Résultats de recherche: Contribution à un journal › Article › Revue par des pairs

Résumé

4-Hydroxy and mercapto pyridines were successfully tested in Ugi-Smiles couplings. Such multicomponent reactions applied to quinoline derivatives afford a very convenient and short synthesis of antimalarial analogues.

langue originale	Anglais
Pages (de - à)	476-478
Nombre de pages	3
journal	Organic Letters
Volume	14
Numéro de publication	2
Les DOIs	https://doi.org/10.1021/ol202974w
état	Publié - 20 janv. 2012
Modification externe	Oui

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10.1021/ol202974w

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title = "Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues",

abstract = "4-Hydroxy and mercapto pyridines were successfully tested in Ugi-Smiles couplings. Such multicomponent reactions applied to quinoline derivatives afford a very convenient and short synthesis of antimalarial analogues.",

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year = "2012",

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journal = "Organic Letters",

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T2 - A fast access to chloroquine analogues

AU - El Kaïm, Laurent

AU - Grimaud, Laurence

AU - Pravin, Patil

PY - 2012/1/20

Y1 - 2012/1/20

N2 - 4-Hydroxy and mercapto pyridines were successfully tested in Ugi-Smiles couplings. Such multicomponent reactions applied to quinoline derivatives afford a very convenient and short synthesis of antimalarial analogues.

AB - 4-Hydroxy and mercapto pyridines were successfully tested in Ugi-Smiles couplings. Such multicomponent reactions applied to quinoline derivatives afford a very convenient and short synthesis of antimalarial analogues.

U2 - 10.1021/ol202974w

DO - 10.1021/ol202974w

M3 - Article

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SN - 1523-7060

VL - 14

SP - 476

EP - 478

JO - Organic Letters

JF - Organic Letters

IS - 2

ER -

Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues

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